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Results for "

nAChR inhibitor

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    79
    TargetMol | Inhibitors_Agonists
  • Peptide Products
    5
    TargetMol | Peptide_Products
  • Dye Reagents
    1
    TargetMol | Dye_Reagents
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    19
    TargetMol | Natural_Products
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    1
    TargetMol | Disease_Modeling_Products
Urethane
Ethylurethane, Ethyl carbamate, Carbamic acid ethyl ester
T005151-79-6
Urethane (Ethylurethane) was an antineoplastic agent .Now is used for other medicinal purposes.
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Galanthamine hydrobromide
Galanthamine HBr, Galantamine hydrobromide
T00861953-04-4
Galanthamine hydrobromide (Galantamine hydrobromide), a long-acting and centrally active AChE inhibitor (IC50:410 nM), is an allosteric potentiator at neuronal nicotinic ACh receptors.
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Cytisinicline
Sophorine, Cytisine, Baptitoxine, Baphitoxine
T0479485-35-8
Cytisinicline (Sophorine), an alkaloid, is found naturally in several plants.
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Choline chloride
Hepacholine, Biocoline, Biocolina
T103967-48-1
Choline chloride (Biocoline) is a basic constituent of lecithin that is found in many plants and animal organs. It is important as a precursor of acetylcholine, as a methyl donor in various metabolic processes, and in lipid metabolism.
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Acetylcholine chloride
ACh chloride, Pilofrin
T122160-31-1
Acetylcholine Chloride is the chloride salt form of acetylcholine, a synthetic, quaternary amino alcohol with cholinergic properties. Acetylcholine chloride (Pilofrin) mimics the parasympathomimetic effect of the endogenous compound acetylcholine. Administered as an ophthalmic solution, this drug stimulates the cholinoceptors in the sphincter muscle of the iris, causing the pupil to constrict.
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(R,S)-Anatabine
T138572743-90-0
(R,S)-Anatabine is a minor tobacco alkaloid found in the Solanaceae family of plants, and serves as a specific marker for detecting tobacco use.
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Arecoline hydrobromide
Arecoline HBr, Arecoline bromide
T2198300-08-3
Arecoline hydrobromide (Arecoline HBr) is a muscarinic acetylcholine receptor agonist.
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(+)-Sparteine
Pachycarpine
T7853492-08-0
(+)-Sparteine ​​is a quinoline alkaloid extracted from Scotch broom, a sodium channel blocker and a class 1a antiarrhythmic agent. It competitively inhibits the activity of nicotinic acetylcholine receptors in nerve cells and is a ganglionic blocking agent.
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Cholesterol myristate
Cholesteryl tetradecanoate, Cholesteryl myristate
T80401989-52-2
Cholesterol Myristate (Cholesteryl Myristate) is a natural steroid found in traditional Chinese medicine that interacts with various ion channels, including the GABAA receptor, nicotinic acetylcholine receptor, and the inward-rectifier potassium ion channel.
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Spinosad
T9076168316-95-8
Spinosad is a naturally-occurring insecticide found in the the soil bacterium S. spinosa. It is a mixture of the macrocyclic lactones spinosyn A and spinosyn D, which act as agonists of insect nicotinic acetylcholinesterase receptors (nAChRs).
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Vinblastine sulfate
NSC49842, Vincaleukoblastine sulfate salt
T1668143-67-9
Vinblastine sulfate (Vincaleukoblastine sulfate salt) can inhibit the formation of microtubule, it also inhibits nAChR(IC50=8.9 uM).
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Catharanthine
(+)-3, 4-Didehydrocoronaridine, (+)-3,4-Didehydrocoronaridine
T27822468-21-5
Catharanthine ((+)-3,4-Didehydrocoronaridine) suppresses nicotinic receptor-mediated diaphragm contractions with an IC50 of 59.6 μM.
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7-10 days
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beta-Eudesmol
Beta-Selinenol
T3865473-15-4
beta-Eudesmol (Beta-Selinenol) is a noncompetitive antagonist of nicotinic acetylcholine receptors (nAChRs). It is a sesquiterpene that has been found in a variety of plants, including Cannabis, and has diverse biological activities.
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N-Methylcytisine
Caulophylline
T5S0994486-86-2
1. N-Methylcytisine (Caulophylline)'s nicotinic receptors have high affinity (KD = 5 nM)to nAChR from squid optical ganglia. 2. N-Methylcytisine and N, N-dimethylcytisine did not displace 14C-tubocurarine at a concentration of .1 mM, cytisine was the only effective inhibitor of 14C-tubocurarine specific binding (Ki=7 nM).
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Myosmine
T7671532-12-7
Myosmine is a minor tobacco alkaloid that is structurally related to nicotine.
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(S)-Coclaurine
Coclaurine
TN1519486-39-5
(S)-Coclaurine (Coclaurine) is an antagonist of nAChR isolated from Sarcopetalum harveyanum.
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Ferulamide
4-Hydroxy-3-methoxycinnamide
TN164361012-31-5
Ferulamide (4-Hydroxy-3-methoxycinnamide), a Ferulic acid derivative, shows potent inhibitory activity against arachidonic acid-induced platelet aggregation.
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Anatoxin-a
ATX-a
TN762364285-06-9
Anatoxin-a (ATX-a), a neurotoxic alkaloid, functions as an agonist for the nicotinic acetylcholine receptor (nAChR) and as an inhibitor of Acetylcholinesterase (AChE) [1] [2].
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α-Conotoxin MII
TP2063175735-93-0
α-Conotoxin MII is a highly potent and selective competitive antagonist for α3β2 subunit-containing nicotinic receptors (IC50 = 0.5 - 3.5 nM at α3β2 expressed in Xenopus oocytes). Also potently blocks β3-containing neuronal nicotinic receptors. Displays >
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